产品描述:
SNC 80 is a selective nonpeptide agonist of the δ-opioid receptor (Ki = 0.18 nM, IC50 = 2.73 nM) that is over 2,000-fold less effective at the μ-opioid receptor.{25516,25513,25515} It effectively activates µ/δ receptor heteromers (EC50 = 52.8 nM) but not κ/δ or μ/κ heteromers.{25524} SNC 80 has antinociceptive as well as pro-convulsant effects in vivo.{25516,25513,25514}