产品描述:
GW 405833 is a partial agonist of the cannabinoid CB2 receptor (EC50 = 0.65 nM).{16338} It is selective for CB2, binding with a Ki value of 14 nM compared to that of CB1 with a Ki value of 2.04 µM.{16338} GW 405833 demonstrates anti-inflammatory and antihyperalgesic properties in animal models of inflammation and pain.{16338}