产品描述:
Carbetapentane is a sigma-1 (σ1) receptor agonist (Ki = 10.4 nM).{25816} In vivo, carbetapentane (1-5 mg/kg) inhibits citric acid-induced cough in guinea pigs.{21421} Carbetapentane (12.5 and 25 mg/kg; i.p.) reduces the number of seizures, mortality, and hippocampal neuronal cell death in a rat model of kainate-induced seizures.{62541}